Composite
68%
Novelty
75%
Feasibility
60%
Impact
83%
Mechanistic
86%
Druggability
Safety
Confidence
48%

Mechanistic description

Symmetric dimethylation of arginine residues in the FUS RGG1/RGG2 domains by PRMT5/PRMT1 maintains FUS in a dynamic liquid phase-separated state by reducing inter-molecular beta-sheet propensity. ALS-linked mutations near the RGG domains reduce arginine methylation efficiency, shifting FUS toward an aggregation-prone unmethylated state. PRMT5 activator treatment in FUS-ALS iPSC motor neurons should restore arginine methylation stoichiometry and increase the concentration required for pathological aggregation by >3-fold.

Evidence for (5)

  • ALS-FUS mutations cause abnormal PARylation and histone H1.2 interaction, leading to pathological changes.

    PMID:39167487 2024 Cell Rep
  • ALS-associated FUS mutation reshapes the RNA and protein composition of stress granules.

    PMID:39494508 2024 Nucleic Acids Res
  • A Liquid-to-Solid Phase Transition of the ALS Protein FUS Accelerated by Disease Mutation.

    PMID:26317470 2015 Cell
  • M6A-dependent RNA condensation underlies FUS autoregulation and can be harnessed for ALS therapy development.

    PMID:40700505 2025 Sci Adv
  • Pathogenesis of FUS-associated ALS and FTD: insights from rodent models.

    PMID:27600654 2016 Acta Neuropathol Commun

Evidence against (2)